Figure 2. ERβ activity at the E-cadherin promoter in PCa cells.
(A) In a redox neutral milieu, ligand binds ERβ and initiates receptor dimerization, occupancy of its cognate DNA-binding element in the E-cadherin promoter, and activation of transcription. (B) In the presence of H2O2, ERβ is oxidized at the 2nd zinc-finger motif and is unable to dimerize, thus destabilizing its DNA-binding capacity and leading to a loss of E-cadherin transcriptional activation.